Chemistry 9701 · AS & A Level · States of matter

States of matter — practice question

Statins are a class of drugs that reduce the level of cholesterol in the blood. Atorvastatin is a statin that is commonly prescribed.
(a(i))[1]

Statins may decompose in the acid present in the stomach. Draw a line through the bond in the atorvastatin structure in Fig. 5.1 that could be cleaved under acidic conditions.

(a(ii))[1]

Use the structure to explain why atorvastatin dissolves in water.

(a(iii))[1]

Complete the molecular formula of atorvastatin. $\text{C H}_{35}\text{N O F}$

(a(iv))[1]

Atorvastatin includes chiral carbon atoms. Circle every chiral carbon atom in Fig. 5.1.

(a(v))[1]

The synthetic preparation of atorvastatin requires the production of a single optical isomer. Suggest why.

(b(i))[1]

The proton ($^1\text{H}$) NMR spectrum of atorvastatin dissolved in $\text{CDCl}_3$ is recorded. Use Table 5.1 to work out the number of hydrogen atoms that could give peaks in the region $\delta = 6.5-13.0$ ppm.

(b(ii))[2]

The proton ($^1\text{H}$) NMR spectrum of atorvastatin dissolved in $\text{D}_2\text{O}$ is recorded. Predict how many hydrogen atoms would not show a peak in this spectrum. Explain your answer.

(c)[2]

Atorvastatin reacts with an excess of $\text{LiAlH}_4$. Name all the functional groups in atorvastatin that react with $\text{LiAlH}_4$. Name the new functional group that would be formed in each case.

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